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FTI 277 hydrochloride
CAS No. 180977-34-8
FTI 277 hydrochloride ( —— )
产品货号. M17384 CAS No. 180977-34-8
FTI 277 hydrochloride is an effective and specific farnesyltransferase (FTase) inhibitor (IC50: 500 pM); this selectivity is about 100-fold than the closely related GGTase I.
纯度: 98%
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 2MG | ￥543 | 有现货 |
|
| 5MG | ￥786 | 有现货 |
|
| 10MG | ￥1499 | 有现货 |
|
| 25MG | ￥2730 | 有现货 |
|
| 50MG | ￥4577 | 有现货 |
|
| 100MG | ￥6423 | 有现货 |
|
| 200MG | 获取报价 | 有现货 |
|
| 500MG | 获取报价 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称FTI 277 hydrochloride
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述FTI 277 hydrochloride is an effective and specific farnesyltransferase (FTase) inhibitor (IC50: 500 pM); this selectivity is about 100-fold than the closely related GGTase I.
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产品描述FTI 277 hydrochloride is an effective and specific farnesyltransferase (FTase) inhibitor (IC50: 500 pM); this selectivity is about 100-fold than the closely related GGTase I.
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同义词——
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通路Angiogenesis
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靶点VEGFR
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受体Farnesyl transferase (FTase); GGTase I
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研究领域Cancer
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适应症——
化学信息
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CAS Number180977-34-8
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分子量484.07
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分子式C22H30ClN3O3S2
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纯度98%
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溶解度DMSO : ≥ 4.9 mg/mL; 10.12 mM
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SMILESCOC(=O)[C@H](CCSC)NC(=O)c1c(cc(cc1)NC[C@H](CS)N)c1ccccc1.Cl
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1. Lerner EC, et al. J Biol Chem. 1995, 270(45), 26802-26806.
产品手册
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